BDBM50238941 CHEMBL4068969

SMILES Cc1cccc(Oc2cccc(COc3ccccc3CCC(=O)OCCCOP(O)(=O)OC[C@H](N)C(O)=O)c2)c1

InChI Key InChIKey=SJODWDYPTIHSMK-UHFFFAOYSA-N

Data  4 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 50238941   

TargetProbable G-protein coupled receptor 34(Mouse)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50238941(CHEMBL4068969)
Affinity DataEC50:  550nMAssay Description:Agonist activity at mouse GPR34 expressed in HEK293 cells co-transfected with AP-TGFalpha/chimeric Galphaq/i1 assessed as induction of ectodomain she...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2019
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 34(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50238941(CHEMBL4068969)
Affinity DataEC50:  230nMAssay Description:Agonist activity at human GPR34 expressed in HEK293 cells co-transfected with AP-TGFalpha/chimeric Galphaq/i1 assessed as induction of AP-TGFalpha re...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2019
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 34(Human)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50238941(CHEMBL4068969)
Affinity DataEC50:  229nMAssay Description:Agonist activity at human GPR34 expressed in HEK293 cells co-transfected with AP-TGFalpha/chimeric Galphaq/i1 assessed as induction of AP-TGFalpha re...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2019
Entry Details Article
PubMed
TargetProbable G-protein coupled receptor 34(Mouse)
The University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50238941(CHEMBL4068969)
Affinity DataEC50:  550nMAssay Description:Agonist activity at mouse GPR34 expressed in HEK293 cells co-transfected with AP-TGFalpha/chimeric Galphaq/i1 assessed as induction of ectodomain she...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2019
Entry Details Article
PubMed