BDBM50238747 CHEMBL4064809

SMILES COc1ccc(F)cc1C1CC1CNCc1ccccc1C#N

InChI Key InChIKey=QOLLBJICSQQCLT-UHFFFAOYSA-N

Data  6 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 6 hits for monomerid = 50238747   

Target5-hydroxytryptamine receptor 2C(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50238747(CHEMBL4064809)
Affinity DataEC50:  245nMAssay Description:Agonist activity at tTA containing TEV cleavage site-fused 5-HT2C-INI receptor isoform (unknown origin) expressed in TEV-fused beta-arrestin2 express...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/11/2019
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50238747(CHEMBL4064809)
Affinity DataEC50:  721nMAssay Description:Agonist activity at human 5-HT2A receptor expressed in Flp-IN HEK293 cells assessed as induction of calcium flux measured every second for 5 mins by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/11/2019
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50238747(CHEMBL4064809)
Affinity DataEC50:  724nMAssay Description:Agonist activity at human 5-HT2A receptor expressed in Flp-IN HEK293 cells assessed as induction of calcium flux measured every second for 5 mins by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/11/2019
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50238747(CHEMBL4064809)
Affinity DataEC50:  238nMAssay Description:Agonist activity at human 5-HT2B receptor expressed in Flp-IN HEK293 cells assessed as induction of calcium flux measured every second for 5 mins by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/11/2019
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2B(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50238747(CHEMBL4064809)
Affinity DataEC50:  240nMAssay Description:Agonist activity at human 5-HT2B receptor expressed in Flp-IN HEK293 cells assessed as induction of calcium flux measured every second for 5 mins by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/11/2019
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50238747(CHEMBL4064809)
Affinity DataEC50:  245nMAssay Description:Agonist activity at human 5-HT2C-INI receptor isoform expressed in Flp-IN HEK293 cells assessed as induction of Gq-mediated calcium flux measured eve...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/11/2019
Entry Details Article
PubMed