BDBM50238308 CHEMBL4103605

SMILES Cc1n[nH]c2nccc(-c3ccc(NC(=O)Nc4cccc(C)c4)cc3)c12

InChI Key InChIKey=GIODDBAYPWNJIQ-UHFFFAOYSA-N

Data  8 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 8 hits for monomerid = 50238308   

TargetPlatelet-derived growth factor receptor alpha(Human)
East China University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50238308(CHEMBL4103605)
Affinity DataIC50: 40nMAssay Description:Inhibition of PDGFRalpha (unknown origin) using FAM-labeled peptide as substrate preincubated for 10 mins followed by substrate addition in presence ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2019
Entry Details Article
PubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
East China University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50238308(CHEMBL4103605)
Affinity DataIC50: 1.88E+3nMAssay Description:Inhibition of FLT3 (unknown origin) using FAM-labeled peptide as substrate preincubated for 10 mins followed by substrate addition in presence of ATP...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2019
Entry Details Article
PubMed
TargetFibroblast growth factor receptor 1(Human)
East China University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50238308(CHEMBL4103605)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of FGFR1 (unknown origin) using FAM-labeled peptide as substrate preincubated for 10 mins followed by substrate addition in presence of AT...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2019
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
East China University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50238308(CHEMBL4103605)
Affinity DataIC50: 1.23E+3nMAssay Description:Inhibition of VEGFR2 (unknown origin) using FAM-labeled peptide as substrate preincubated for 10 mins followed by substrate addition in presence of A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2019
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 1(Human)
East China University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50238308(CHEMBL4103605)
Affinity DataIC50: 3.49E+3nMAssay Description:Inhibition of VEGFR1 (unknown origin) using FAM-labeled peptide as substrate preincubated for 10 mins followed by substrate addition in presence of A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2019
Entry Details Article
PubMed
TargetMast/stem cell growth factor receptor Kit(Human)
East China University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50238308(CHEMBL4103605)
Affinity DataIC50: 2.10nMAssay Description:Inhibition of cKIT (unknown origin) using FAM-labeled peptide as substrate preincubated for 10 mins followed by substrate addition in presence of ATP...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2019
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 3(Human)
East China University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50238308(CHEMBL4103605)
Affinity DataIC50: 376nMAssay Description:Inhibition of VEGFR3 (unknown origin) using FAM-labeled peptide as substrate preincubated for 10 mins followed by substrate addition in presence of A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2019
Entry Details Article
PubMed
TargetPlatelet-derived growth factor receptor beta(Human)
East China University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50238308(CHEMBL4103605)
Affinity DataIC50: 197nMAssay Description:Inhibition of PDGFRbeta (unknown origin) using FAM-labeled peptide as substrate preincubated for 10 mins followed by substrate addition in presence o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2019
Entry Details Article
PubMed