BDBM50233007 CHEMBL403139::N-((1S,13bR)-6-chloro-1,2,3,4,9,13b-hexahydro-4a-aza-tribenzo[a,c,e]cyclohepten-1-yl)-2,2,2-trifluoro-acetamide

SMILES FC(F)(F)C(=O)N[C@H]1CCCN2[C@@H]1c1ccccc1Cc1ccc(Cl)cc21

InChI Key InChIKey=HAXRSFLRCIBMMN-UHFFFAOYSA-N

Data  1 IC50  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50233007   

TargetProgesterone receptor(Human)
Nv Organon

Curated by ChEMBL
LigandPNGBDBM50233007(N-((1S,13bR)-6-chloro-1,2,3,4,9,13b-hexahydro-4a-a...)
Affinity DataIC50: 26nMAssay Description:Inhibition of progesterone receptor expressed in CHO cells by luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetProgesterone receptor(Human)
Nv Organon

Curated by ChEMBL
LigandPNGBDBM50233007(N-((1S,13bR)-6-chloro-1,2,3,4,9,13b-hexahydro-4a-a...)
Affinity DataEC50:  2nMAssay Description:Agonist activity at progesterone receptor expressed in CHO cells by luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed