BDBM50232142 1-(1H-indazol-4-yl)-3-(1-(4-(trifluoromethyl)phenyl)ethyl)urea::CHEMBL397922

SMILES CC(NC(=O)Nc1cccc2[nH]ncc12)c1ccc(cc1)C(F)(F)F

InChI Key InChIKey=SLVGTOOOMMCFEW-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50232142   

LigandPNGBDBM50232142(1-(1H-indazol-4-yl)-3-(1-(4-(trifluoromethyl)pheny...)
Affinity DataIC50: 47nMAssay Description:Blockade of human TRPV1 receptor assessed as inhibition of capsaicin-induced calcium fluxMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
LigandPNGBDBM50232142(1-(1H-indazol-4-yl)-3-(1-(4-(trifluoromethyl)pheny...)
Affinity DataIC50: 47nMAssay Description:Antagonist activity at human TRPV1 assessed as inhibition of calcium influxMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed