BDBM50232120 1-(1H-indazol-4-yl)-3-(4-(pyrrolidin-1-yl)-2,3-dihydro-1H-inden-1-yl)urea::CHEMBL399434

SMILES O=C(NC1CCc2c1cccc2N1CCCC1)Nc1cccc2[nH]ncc12

InChI Key InChIKey=UOHCGMBECWOBEU-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50232120   

TargetTransient receptor potential cation channel subfamily V member 1(Human)
Abbott Laboratories

Curated by ChEMBL

LigandBDBM50232120(1-(1H-indazol-4-yl)-3-(4-(pyrrolidin-1-yl)-2,3-dih...)Copy SMILESCopy InChI

Affinity DataIC50: 21nMAssay Description:Blockade of human TRPV1 receptor assessed as inhibition of capsaicin-induced calcium fluxMore data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In Depth
Date in BDB:
11/11/2009
Entry Details Article
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