BDBM50232119 1-(5-methoxy-2,3-dihydro-1H-inden-1-yl)-3-(1H-indazol-4-yl)urea::CHEMBL430402

SMILES COc1ccc2C(CCc2c1)NC(=O)Nc1cccc2[nH]ncc12

InChI Key InChIKey=ZBISBOUCIVCJOF-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50232119   

TargetTransient receptor potential cation channel subfamily V member 1(Human)
Abbott Laboratories

Curated by ChEMBL

LigandBDBM50232119(1-(5-methoxy-2,3-dihydro-1H-inden-1-yl)-3-(1H-inda...)Copy SMILESCopy InChI

Affinity DataIC50: 40nMAssay Description:Blockade of human TRPV1 receptor assessed as inhibition of capsaicin-induced calcium fluxMore data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In Depth
Date in BDB:
11/11/2009
Entry Details Article
Copy Entry DOIPubMed
Copy Rxn URL