BDBM50231119 CHEMBL254877::N-(2-(5-methoxy-1H-indol-3-yl)ethyl)-4-(1,1,2,2-tetrafluoroethoxy)benzamide

SMILES COc1ccc2[nH]cc(CCNC(=O)c3ccc(OC(F)(F)C(F)F)cc3)c2c1

InChI Key InChIKey=AIGNOHAPRJHNHK-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50231119   

TargetTransient receptor potential cation channel subfamily V member 1(Human)
Pfizer

Curated by ChEMBL

LigandBDBM50231119(N-(2-(5-methoxy-1H-indol-3-yl)ethyl)-4-(1,1,2,2-te...)Copy SMILESCopy InChI

Affinity DataIC50: 1.64E+3nMAssay Description:Antagonist activity at human TRPV1 assessed as inhibition of capsaicin-induced calcium influx in HEK293 cellsMore data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In Depth
Date in BDB:
11/11/2009
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