BDBM50231114 CHEMBL254048::N-(1-(6-hydroxyquinolin-4-yl)propan-2-yl)-4-(trifluoromethoxy)benzamide

SMILES CC(Cc1ccnc2ccc(O)cc12)NC(=O)c1ccc(OC(F)(F)F)cc1

InChI Key InChIKey=QDMYIDQIFWFEIY-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50231114   

TargetTransient receptor potential cation channel subfamily V member 1(Human)
Pfizer

Curated by ChEMBL

LigandBDBM50231114(N-(1-(6-hydroxyquinolin-4-yl)propan-2-yl)-4-(trifl...)Copy SMILESCopy InChI

Affinity DataIC50: 740nMAssay Description:Antagonist activity at human TRPV1 assessed as inhibition of capsaicin-induced calcium influx in HEK293 cellsMore data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In Depth
Date in BDB:
11/11/2009
Entry Details Article
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