BDBM50231085 CHEMBL254905::N-(2,4-dichlorophenethyl)-4-(trifluoromethoxy)benzamide

SMILES FC(F)(F)Oc1ccc(cc1)C(=O)NCCc1ccc(Cl)cc1Cl

InChI Key InChIKey=OFTCRLPSTWMOTG-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50231085   

TargetTransient receptor potential cation channel subfamily V member 1(Human)
Pfizer

Curated by ChEMBL

LigandBDBM50231085(N-(2,4-dichlorophenethyl)-4-(trifluoromethoxy)benz...)Copy SMILESCopy InChI

Affinity DataIC50: 2.56E+3nMAssay Description:Antagonist activity at human TRPV1 assessed as inhibition of capsaicin-induced calcium influx in HEK293 cellsMore data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In Depth
Date in BDB:
11/11/2009
Entry Details Article
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