BDBM50231068 CHEMBL252782::N-(4-tert-butylphenyl)-4-(trifluoromethyl)benzamide

SMILES CC(C)(C)c1ccc(NC(=O)c2ccc(cc2)C(F)(F)F)cc1

InChI Key InChIKey=HZCDZHJWDCXUHT-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50231068   

TargetTransient receptor potential cation channel subfamily V member 1(Human)
Pfizer

Curated by ChEMBL

LigandBDBM50231068(N-(4-tert-butylphenyl)-4-(trifluoromethyl)benzamid...)Copy SMILESCopy InChI

Affinity DataIC50: 220nMAssay Description:Antagonist activity at human TRPV1 assessed as inhibition of capsaicin-induced calcium influx in HEK293 cellsMore data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In Depth
Date in BDB:
11/11/2009
Entry Details Article
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