BDBM50229938 CHEMBL1592888

SMILES Cc1c(C(=O)c2cccc3ccccc23)c2cccc3OC[C@H](CN4CCOCC4)n1c23

InChI Key InChIKey=HQVHOQAKMCMIIM-UHFFFAOYSA-N

Data  1 IC50  2 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 50229938   

TargetCannabinoid receptor 1/2(Rat)
Sterling Research Group

Curated by ChEMBL
LigandPNGBDBM50229938(CHEMBL1592888)
Affinity DataIC50: 8.00E+3nMAssay Description:Concentration required to displace 50% of 0.5 nM [3H](aminoalkyl)indole binding to cannabinoid receptor in rat cerebellum membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/15/2019
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
Curtin University

Curated by ChEMBL
LigandPNGBDBM50229938(CHEMBL1592888)
Affinity DataEC50:  284nMAssay Description:Agonist activity at human CB1R expressed in mouse AtT20 cells by FLIPR membrane potential assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
PubMed
TargetCannabinoid receptor 2(Human)
Curtin University

Curated by ChEMBL
LigandPNGBDBM50229938(CHEMBL1592888)
Affinity DataEC50:  62nMAssay Description:Agonist activity at human CB2R expressed in mouse AtT20 cells by FLIPR membrane potential assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/19/2023
Entry Details
PubMed