BDBM50227753 2-(4-(3-((2,4-bis(trifluoromethyl)benzamido)methyl)phenoxy)-2-methylphenoxy)-2-methylpropanoic acid::CHEMBL237084

SMILES Cc1cc(Oc2cccc(CNC(=O)c3ccc(cc3C(F)(F)F)C(F)(F)F)c2)ccc1OC(C)(C)C(O)=O

InChI Key InChIKey=SOKGUCREKPAHNX-UHFFFAOYSA-N

Data  9 IC50  2 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 11 hits for monomerid = 50227753   

LigandPNGBDBM50227753(2-(4-(3-((2,4-bis(trifluoromethyl)benzamido)methyl...)
Affinity DataEC50:  2.87E+3nMAssay Description:Agonist activity at human PPARdelta expressed in CV1 cells by receptor transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
LigandPNGBDBM50227753(2-(4-(3-((2,4-bis(trifluoromethyl)benzamido)methyl...)
Affinity DataEC50:  1.06E+3nMAssay Description:Agonist activity at human PPARgamma expressed in CV1 cells by receptor transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
LigandPNGBDBM50227753(2-(4-(3-((2,4-bis(trifluoromethyl)benzamido)methyl...)
Affinity DataIC50: 203nMAssay Description:Displacement of [3H]2-methyl-2-(4-{3-{propyl-(5-pyridin-2-yl-thiophene-2-sulfonyl)-amino}-propyl}-phenoxy)-propionic acid from human PPARgammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
LigandPNGBDBM50227753(2-(4-(3-((2,4-bis(trifluoromethyl)benzamido)methyl...)
Affinity DataIC50: 1.03E+4nMAssay Description:Displacement of [3H]2-(4-{2-[3-(2,4-difluoro-phenyl)-1-heptyl-ureido]-ethyl}-phenoxy)-2-methyl-butyric acid from human PPARalphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
LigandPNGBDBM50227753(2-(4-(3-((2,4-bis(trifluoromethyl)benzamido)methyl...)
Affinity DataIC50: 40nMAssay Description:Displacement of [3H]2-(4-{2-[3-(2,4-difluoro-phenyl)-1-heptyl-ureido]-ethyl}-phenoxy)-2-methyl-butyric acid from human PPARdeltaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
LigandPNGBDBM50227753(2-(4-(3-((2,4-bis(trifluoromethyl)benzamido)methyl...)
Affinity DataIC50: 40.0nMAssay Description:Agonist activity at PPARdeltaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
LigandPNGBDBM50227753(2-(4-(3-((2,4-bis(trifluoromethyl)benzamido)methyl...)
Affinity DataIC50: 1.03E+4nMAssay Description:Agonist activity at PPARalphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
LigandPNGBDBM50227753(2-(4-(3-((2,4-bis(trifluoromethyl)benzamido)methyl...)
Affinity DataIC50: 40nMAssay Description:Agonist activity at PPARdeltaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
LigandPNGBDBM50227753(2-(4-(3-((2,4-bis(trifluoromethyl)benzamido)methyl...)
Affinity DataIC50: 203nMAssay Description:Agonist activity at PPARgammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
LigandPNGBDBM50227753(2-(4-(3-((2,4-bis(trifluoromethyl)benzamido)methyl...)
Affinity DataIC50: 1.03E+4nMAssay Description:Agonist activity at PPARalphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
LigandPNGBDBM50227753(2-(4-(3-((2,4-bis(trifluoromethyl)benzamido)methyl...)
Affinity DataIC50: 203nMAssay Description:Agonist activity at PPARgammaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed