BDBM50219939 CHEMBL240693::N-((1r,4r)-4-(2-(4-(2,3-dichlorophenyl)piperazin-1-yl)ethyl)cyclohexyl)pyridine-3-sulfonamide

SMILES Clc1cccc(N2CCN(CC[C@H]3CC[C@@H](CC3)NS(=O)(=O)c3cccnc3)CC2)c1Cl

InChI Key InChIKey=DLCUNIPVNVPKEI-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50219939   

TargetD(2) dopamine receptor(Rat)
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50219939(N-((1r,4r)-4-(2-(4-(2,3-dichlorophenyl)piperazin-1...)
Affinity DataIC50: 4nMAssay Description:Displacement of [3H]spiperone from dopamine D2 receptor in rat striatal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(3) dopamine receptor(Rat)
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50219939(N-((1r,4r)-4-(2-(4-(2,3-dichlorophenyl)piperazin-1...)
Affinity DataIC50: 0.200nMAssay Description:Displacement of [3H]spiperone from rat dopamine D3 receptor expressed in Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed