BDBM50217900 3-(6-chloro-imidazo[2,1-b]thiazole-5-sulfonyl)-1-pyrrolidin-3-yl-1H-pyrrolo[2,3-b]pyridine::CHEMBL236103

SMILES ClC1=NC2SC=CN2C1S(=O)(=O)c1cn(C2CCNC2)c2ncccc12

InChI Key InChIKey=HXUMXEGSBWZJND-UHFFFAOYSA-N

Data  1 KI  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50217900   

Target5-hydroxytryptamine receptor 6(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50217900(3-(6-chloro-imidazo[2,1-b]thiazole-5-sulfonyl)-1-p...)
Affinity DataEC50:  80nMAssay Description:Agonist activity at human 5HT6 expressed in HeLa cells assessed as intracellular cAMP level by radioimmunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50217900(3-(6-chloro-imidazo[2,1-b]thiazole-5-sulfonyl)-1-p...)
Affinity DataKi:  1nMAssay Description:Displacement of [3H]LSD from cloned human 5HT6 expressed in HeLa cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed