BDBM50211536 CHEMBL389891::N-((3R,4S)-6-((S)-2-((2,6-dimethylphenylamino)methyl)pyrrolidine-1-carbonyl)-3-hydroxy-2,2-dimethyl-3,4-dihydro-2H-chromen-4-yl)-4-ethylbenzenesulfonamide

SMILES CCc1ccc(cc1)S(=O)(=O)N[C@@H]1[C@@H](O)C(C)(C)Oc2ccc(cc12)C(=O)N1CCC[C@H]1CNc1c(C)cccc1C

InChI Key InChIKey=ZGNURVKJDROBKC-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50211536   

TargetPotassium voltage-gated channel subfamily A member 5(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50211536(N-((3R,4S)-6-((S)-2-((2,6-dimethylphenylamino)meth...)
Affinity DataIC50: 260nMAssay Description:Inhibition of human Kv1.5 channel expressed in mouse L929 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed