BDBM50211523 (3S,4R)-4-(4-ethyl-N-(pyridin-3-ylmethyl)phenylsulfonamido)-3-hydroxy-2,2-dimethyl-N-phenethylchroman-6-carboxamide::CHEMBL230564

SMILES CCc1ccc(cc1)S(=O)(=O)N(Cc1cccnc1)[C@H]1[C@H](O)C(C)(C)Oc2ccc(cc12)C(=O)NCCc1ccccc1

InChI Key InChIKey=RFJFPAJIZZZGKJ-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50211523   

TargetPotassium voltage-gated channel subfamily A member 5(Human)
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50211523((3S,4R)-4-(4-ethyl-N-(pyridin-3-ylmethyl)phenylsul...)
Affinity DataIC50: 130nMAssay Description:Inhibition of human Kv1.5 channel expressed in mouse L929 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed