BDBM50209693 1-(4-biphenylmethyl)-3-(2-hydroxy-1,1-dimethylethyl)-1-{2-[1-(4-methylbenzyl)-4-piperidinyl]ethyl}urea::CHEMBL240940

SMILES Cc1ccc(CN2CCC(CCN(Cc3ccc(cc3)-c3ccccc3)C(=O)NC(C)(C)CO)CC2)cc1

InChI Key InChIKey=DXTFGJMQKYMFGQ-UHFFFAOYSA-N

Data  2 KI

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Similarity at least:  must be >=0.5
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50209693   

TargetMelanin-concentrating hormone receptor 1(Human)
University of Navarra

Curated by ChEMBL
LigandPNGBDBM50209693(1-(4-biphenylmethyl)-3-(2-hydroxy-1,1-dimethylethy...)
Affinity DataKi:  144nMAssay Description:Displacement of [3H]SNAP from human MCH1 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
University of Navarra

Curated by ChEMBL
LigandPNGBDBM50209693(1-(4-biphenylmethyl)-3-(2-hydroxy-1,1-dimethylethy...)
Affinity DataKi:  144nMAssay Description:Displacement of [3H]SNAP-7941 from human MCHR1 expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed