BDBM50208151 CHEMBL3986483::US9708270, 97

SMILES OC(=O)CC1CCC2(CCN(CC2)c2cc(OC(F)(F)F)ccc2Cl)OC1

InChI Key InChIKey=DIZADOFRCFKNSD-UHFFFAOYSA-N

Data  4 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Similarity at least:  must be >=0.5
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 50208151   

TargetFree fatty acid receptor 4(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50208151(US9708270, 97 | CHEMBL3986483)
Affinity DataEC50:  5.70E+3nMAssay Description:Agonist activity at human GPR120 short isoform expressed in CHOK1 cells assessed as induction of IP1 accumulation after 60 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2018
Entry Details Article
PubMed
TargetFree fatty acid receptor 4(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50208151(US9708270, 97 | CHEMBL3986483)
Affinity DataEC50:  5.70E+3nMAssay Description:Agonist activity at human GPR120 short isoform expressed in CHOK1 cells assessed as induction of IP1 accumulation after 60 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2018
Entry Details Article
PubMed
TargetFree fatty acid receptor 4(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50208151(US9708270, 97 | CHEMBL3986483)
Affinity DataEC50:  2.10E+3nMAssay Description:Agonist activity at ARMS2-PK2 -tagged human GPR120 short isoform expressed in CHOK1 cells assessed as induction of beta-arrestin2 recruitment after 9...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2018
Entry Details Article
PubMed
TargetFree fatty acid receptor 4(Human)
Merck

Curated by ChEMBL
LigandPNGBDBM50208151(US9708270, 97 | CHEMBL3986483)
Affinity DataEC50:  1.29E+3nMAssay Description:On the day before the measurement day, CHO cells expressing human GPR120 were plated at 10000 cells per well in a 384-well black plate (#3702, Cornin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
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