BDBM50207665 CHEMBL3973096

SMILES COc1cc(CN(CC(N)=O)C(=O)c2cccs2)ccc1OCc1ccc(F)cc1

InChI Key InChIKey=IODQTPLMRRQXND-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50207665   

TargetTransient receptor potential cation channel subfamily M member 8(Human)
Kissei Pharmaceutical

Curated by ChEMBL

LigandBDBM50207665(CHEMBL3973096)Copy SMILESCopy InChI

Affinity DataIC50: 9.10E+3nMAssay Description:Antagonist activity at human recombinant TRPM8 expressed in HEK293 cells assessed as inhibition of menthol-induced calcium increase by Fluo-4 AM base...More data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In Depth
Date in BDB:
8/29/2018
Entry Details Article
Copy Entry DOIPubMed
Copy Rxn URL