BDBM50207567 CHEMBL3936873

SMILES COc1cc(CN([C@@H](C(N)=O)c2ccccc2)C(=O)c2cccs2)ccc1OCc1ccc(F)cc1

InChI Key InChIKey=HKYHALFWTFNENI-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50207567   

TargetTransient receptor potential cation channel subfamily M member 8(Human)
Kissei Pharmaceutical

Curated by ChEMBL

LigandBDBM50207567(CHEMBL3936873)Copy SMILESCopy InChI

Affinity DataIC50: 1.00E+5nMAssay Description:Antagonist activity at human recombinant TRPM8 expressed in HEK293 cells assessed as inhibition of menthol-induced calcium increase by Fluo-4 AM base...More data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In Depth
Date in BDB:
8/29/2018
Entry Details Article
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