BDBM50201371 CHEMBL241265::N-(3-chloro-4-(trifluoromethyl)phenyl)-1-methyl-4-(pyridin-4-ylmethylamino)-1H-pyrazole-5-carboxamide

SMILES Cn1ncc(NCc2ccncc2)c1C(=O)Nc1ccc(c(Cl)c1)C(F)(F)F

InChI Key InChIKey=CNWRDLKCPGZLLP-UHFFFAOYSA-N

Data  3 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 50201371   

TargetVascular endothelial growth factor receptor 2(Human)
Chemical Diversity

Curated by ChEMBL
LigandPNGBDBM50201371(N-(3-chloro-4-(trifluoromethyl)phenyl)-1-methyl-4-...)
Affinity DataIC50: 440nMAssay Description:Inhibition of VEGFR2 by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 2(Human)
Chemical Diversity

Curated by ChEMBL
LigandPNGBDBM50201371(N-(3-chloro-4-(trifluoromethyl)phenyl)-1-methyl-4-...)
Affinity DataIC50: 79nMAssay Description:Inhibition of VEGFR2 by cell-based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVascular endothelial growth factor receptor 1(Human)
Chemical Diversity

Curated by ChEMBL
LigandPNGBDBM50201371(N-(3-chloro-4-(trifluoromethyl)phenyl)-1-methyl-4-...)
Affinity DataIC50: 210nMAssay Description:Inhibition of VEGFR1 by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed