BDBM50200497 2-Amino-5H-phenanthridin-6-one::2-aminophenanthridin-6(5H)-one::CHEMBL225725

SMILES Nc1ccc2[nH]c(=O)c3ccccc3c2c1

InChI Key InChIKey=YMTIEBMDXHJRKO-UHFFFAOYSA-N

Data  3 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 50200497   

TargetPoly [ADP-ribose] polymerase 1(Human)
Guilford Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50200497(2-aminophenanthridin-6(5H)-one | 2-Amino-5H-phenan...)
Affinity DataIC50: 180nMAssay Description:Inhibitory concentration against purified recombinant human poly (ADP-ribose) polymerase-1 (PARP1)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/3/2012
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50200497(2-aminophenanthridin-6(5H)-one | 2-Amino-5H-phenan...)
Affinity DataIC50: 2.67E+5nMAssay Description:Inhibition of HIV1 integrase strand transfer activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50200497(2-aminophenanthridin-6(5H)-one | 2-Amino-5H-phenan...)
Affinity DataIC50: 2.06E+5nMAssay Description:Inhibition of HIV1 integrase 3'-end processing activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2020
Entry Details Article
PubMed