BDBM50199236 6-(4-chlorophenyl)-3-{2-[(4-methyl-1-piperazinyl)methyl]-6-quinolinyl}thieno[3,2-d]pyrimidin-4(3H)-one::CHEMBL214808

SMILES CN1CCN(Cc2ccc3cc(ccc3n2)-n2cnc3cc(sc3c2=O)-c2ccc(Cl)cc2)CC1

InChI Key InChIKey=YLNMKOAPZKIZAU-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50199236   

TargetPotassium voltage-gated channel subfamily H member 2(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50199236(6-(4-chlorophenyl)-3-{2-[(4-methyl-1-piperazinyl)m...)
Affinity DataIC50: 2.19E+4nMAssay Description:Inhibitory activity against hERG by patch-clamp assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50199236(6-(4-chlorophenyl)-3-{2-[(4-methyl-1-piperazinyl)m...)
Affinity DataIC50: 3.10nMAssay Description:Antagonist activity against human MCHR1 expressed in CHO cells by Gal4/Elk1-Luc reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed