BDBM50195077 2-methoxy-2-methyl-3-(5-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)pyridin-2-yl)propanoic acid::CHEMBL222121

SMILES COC(C)(Cc1ccc(OCCc2nc(oc2C)-c2ccccc2)cn1)C(O)=O

InChI Key InChIKey=HLEQAMRJYWQJCX-UHFFFAOYSA-N

Data  2 KI  2 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 50195077   

LigandPNGBDBM50195077(2-methoxy-2-methyl-3-(5-(2-(5-methyl-2-phenyloxazo...)
Affinity DataEC50:  335nMAssay Description:Agonist activity at human PPAR gamma in HepG2 cells by PPAR-GAL4 transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50195077(2-methoxy-2-methyl-3-(5-(2-(5-methyl-2-phenyloxazo...)
Affinity DataEC50:  882nMAssay Description:Agonist activity at human PPAR alpha in HepG2 cells by PPAR-GAL4 transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50195077(2-methoxy-2-methyl-3-(5-(2-(5-methyl-2-phenyloxazo...)
Affinity DataKi:  1.60E+3nMAssay Description:Displacement of radiolabeled darglitazone from human PPAR gamma by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50195077(2-methoxy-2-methyl-3-(5-(2-(5-methyl-2-phenyloxazo...)
Affinity DataKi:  4.80E+3nMAssay Description:Displacement of radiolabeled GW-2331 from human PPAR alpha by SPA assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed