BDBM50194975 2-methoxy-2-methyl-3-(6-(2-(5-methyl-2-phenyloxazol-4-yl)ethoxy)pyridin-3-yl)propanoic acid::CHEMBL221850

SMILES COC(C)(Cc1ccc(OCCc2nc(oc2C)-c2ccccc2)nc1)C(O)=O

InChI Key InChIKey=QQJHRCMKKXNPSH-UHFFFAOYSA-N

Data  1 KI  3 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 50194975   

LigandPNGBDBM50194975(2-methoxy-2-methyl-3-(6-(2-(5-methyl-2-phenyloxazo...)
Affinity DataEC50:  232nMAssay Description:Agonist activity at human PPAR gamma in a HepG2 cells by PPAR-GAL4 transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50194975(2-methoxy-2-methyl-3-(6-(2-(5-methyl-2-phenyloxazo...)
Affinity DataEC50:  144nMAssay Description:Agonist activity at human PPAR alpha in a HepG2 cells by PPAR-GAL4 transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50194975(2-methoxy-2-methyl-3-(6-(2-(5-methyl-2-phenyloxazo...)
Affinity DataEC50:  330nMAssay Description:Displacement of radiolabeled GW-2331 from human PPAR alpha by SPA binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50194975(2-methoxy-2-methyl-3-(6-(2-(5-methyl-2-phenyloxazo...)
Affinity DataKi:  560nMAssay Description:Displacement of radiolabeled darglitazone from human PPAR gamma by SPA binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed