BDBM50194973 2-((6-(2-(2-(4-cyanophenyl)-5-methyloxazol-4-yl)ethoxy)pyridin-3-yl)methyl)-tetrahydrofuran-2-carboxylic acid::CHEMBL217907

SMILES Cc1oc(nc1CCOc1ccc(CC2(CCCO2)C(O)=O)cn1)-c1ccc(cc1)C#N

InChI Key InChIKey=YWXSUMRZNARHPW-UHFFFAOYSA-N

Data  1 KI  3 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 50194973   

LigandPNGBDBM50194973(2-((6-(2-(2-(4-cyanophenyl)-5-methyloxazol-4-yl)et...)
Affinity DataEC50:  31nMAssay Description:Agonist activity at human PPAR alpha in a HepG2 cells by PPAR-GAL4 transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50194973(2-((6-(2-(2-(4-cyanophenyl)-5-methyloxazol-4-yl)et...)
Affinity DataEC50:  28nMAssay Description:Agonist activity at human PPAR gamma in a HepG2 cells by PPAR-GAL4 transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50194973(2-((6-(2-(2-(4-cyanophenyl)-5-methyloxazol-4-yl)et...)
Affinity DataEC50:  314nMAssay Description:Displacement of radiolabeled GW-2331 from human PPAR alpha by SPA binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50194973(2-((6-(2-(2-(4-cyanophenyl)-5-methyloxazol-4-yl)et...)
Affinity DataKi:  334nMAssay Description:Displacement of radiolabeled darglitazone from human PPAR gamma by SPA binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed