BDBM50193598 CHEMBL386043::Dhp-c[D-Cys-Gly-Phe(pNO2)-D-Cys]NH2

SMILES Cc1cc(O)cc(C)c1CCC(=O)N[C@H]1CSSC[C@H](NC(=O)[C@H](Cc2ccc(cc2)[N+]([O-])=O)NC(=O)CNC1=O)C(N)=O

InChI Key InChIKey=UHOUPDXHBXXBLE-UHFFFAOYSA-N

Data  3 KI

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 50193598   

TargetMu-type opioid receptor(Rat)
National University of Singapore

Curated by ChEMBL
LigandPNGBDBM50193598(Dhp-c[D-Cys-Gly-Phe(pNO2)-D-Cys]NH2 | CHEMBL386043)
Affinity DataKi:  4.79nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
National University of Singapore

Curated by ChEMBL
LigandPNGBDBM50193598(Dhp-c[D-Cys-Gly-Phe(pNO2)-D-Cys]NH2 | CHEMBL386043)
Affinity DataKi:  11.6nMAssay Description:Displacement of [3H]DSLET from delta opioid receptor in rat brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
National University of Singapore

Curated by ChEMBL
LigandPNGBDBM50193598(Dhp-c[D-Cys-Gly-Phe(pNO2)-D-Cys]NH2 | CHEMBL386043)
Affinity DataKi:  299nMAssay Description:Displacement of [3H]U-69593 from kappa opioid receptor in guinea pig brain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed