BDBM50191053 1-ethyl-3-(3-oxo-3-((1-phenethylpiperidin-4-yl)(phenyl)amino)propyl)urea::CHEMBL385909

SMILES CCNC(=O)NCCC(=O)N(C1CCN(CCc2ccccc2)CC1)c1ccccc1

InChI Key InChIKey=JFWGDNMHRRUUTG-UHFFFAOYSA-N

Data  3 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 50191053   

TargetDelta-type opioid receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50191053(1-ethyl-3-(3-oxo-3-((1-phenethylpiperidin-4-yl)(ph...)
Affinity DataIC50: 6.65E+3nMAssay Description:Displacement of [3H]DPDPE from human delta opioid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50191053(1-ethyl-3-(3-oxo-3-((1-phenethylpiperidin-4-yl)(ph...)
Affinity DataIC50: 30nMAssay Description:Displacement of [3H]DAMGO from rat mu opioid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50191053(1-ethyl-3-(3-oxo-3-((1-phenethylpiperidin-4-yl)(ph...)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of mu opioid receptor in guinea pig ileum assessed as inhibition of electrically-stimulated muscle contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article
PubMed