BDBM50189293 CHEMBL3827279

SMILES CCOC(=O)c1cc(C(=O)\C=C\c2ccc3N(C)c4ccccc4Sc3c2)n2c(C)cccc12

InChI Key InChIKey=UOZSXSDLAGEQQS-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50189293   

TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Human)
Alexandru Ioan Cuza University

Curated by ChEMBL

LigandBDBM50189293(CHEMBL3827279)Copy SMILESCopy InChI

Affinity DataIC50: 23nMAssay Description:Inhibition of human recombinant farnesyltransferase using farnesylpyrophosphate and dansyl-GCVLS as substrate measured for 15 mins by fluorescence as...More data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In Depth
Date in BDB:
10/11/2017
Entry Details Article
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