BDBM50184747 2-(4-(trifluoromethyl)phenyl)-1,2-dihydroindazol-3-one::CHEMBL3144796

SMILES FC(F)(F)c1ccc(cc1)-n1[nH]c2ccccc2c1=O

InChI Key InChIKey=XQRFOKRJVHIBPI-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50184747   

TargetTransient receptor potential cation channel subfamily V member 1(Human)
Merck Sharp & Dohme

Curated by ChEMBL

LigandBDBM50184747(2-(4-(trifluoromethyl)phenyl)-1,2-dihydroindazol-3...)Copy SMILESCopy InChI

Affinity DataIC50: 340nMAssay Description:Antagonist activity against capsaicin-induced intracellular calcium ion increase in CHO cells expressing human TRPV1 in FLIPR assayMore data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In Depth
Date in BDB:
11/10/2009
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