BDBM50184742 2-(4-tert-butylphenyl)-6-(3-(trifluoromethyl)pyridin-2-yl)-1H-benzo[d]imidazole::CHEMBL211051

SMILES CC(C)(C)c1ccc(cc1)-c1nc2cc(ccc2[nH]1)-c1ncccc1C(F)(F)F

InChI Key InChIKey=CZXZLJJJPXAZQU-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50184742   

TargetTransient receptor potential cation channel subfamily V member 1(Human)
Merck Sharp & Dohme

Curated by ChEMBL

LigandBDBM50184742(2-(4-tert-butylphenyl)-6-(3-(trifluoromethyl)pyrid...)Copy SMILESCopy InChI

Affinity DataIC50: 224nMAssay Description:Antagonist activity against capsaicin-induced intracellular calcium ion increase in CHO cells expressing human TRPV1 in FLIPR assayMore data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In Depth
Date in BDB:
11/10/2009
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