BDBM50184740 6-(3-methylpyridin-2-yl)-2-(4-(trifluoromethyl)phenyl)-1,2-dihydroindazol-3-one::CHEMBL3144707

SMILES Cc1cccnc1-c1ccc2c(c1)[nH]n(-c1ccc(cc1)C(F)(F)F)c2=O

InChI Key InChIKey=NDCDEIBRKPCRDY-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50184740   

TargetTransient receptor potential cation channel subfamily V member 1(Human)
Merck Sharp & Dohme

Curated by ChEMBL

LigandBDBM50184740(6-(3-methylpyridin-2-yl)-2-(4-(trifluoromethyl)phe...)Copy SMILESCopy InChI

Affinity DataIC50: 180nMAssay Description:Antagonist activity against capsaicin-induced intracellular calcium ion increase in CHO cells expressing human TRPV1 in FLIPR assayMore data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In Depth
Date in BDB:
11/10/2009
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