BDBM50184733 CHEMBL210667::N-(4-(3-methylpyridin-2-yl)phenyl)-3-(trifluoromethyl)benzamide

SMILES Cc1cccnc1-c1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1

InChI Key InChIKey=MKXNDOBTTLYFNU-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50184733   

TargetTransient receptor potential cation channel subfamily V member 1(Human)
Merck Sharp & Dohme

Curated by ChEMBL

LigandBDBM50184733(N-(4-(3-methylpyridin-2-yl)phenyl)-3-(trifluoromet...)Copy SMILESCopy InChI

Affinity DataIC50: 640nMAssay Description:Antagonist activity against capsaicin-induced intracellular calcium ion increase in CHO cells expressing human TRPV1 in FLIPR assayMore data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In Depth
Date in BDB:
11/10/2009
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