BDBM50184731 6-(2-methoxyphenyl)-2-(4-(trifluoromethyl)phenyl)-1,2-dihydroindazol-3-one::CHEMBL3144797

SMILES COc1ccccc1-c1ccc2c(c1)[nH]n(-c1ccc(cc1)C(F)(F)F)c2=O

InChI Key InChIKey=DINMMAYTUYCAMR-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50184731   

TargetTransient receptor potential cation channel subfamily V member 1(Human)
Merck Sharp & Dohme

Curated by ChEMBL

LigandBDBM50184731(6-(2-methoxyphenyl)-2-(4-(trifluoromethyl)phenyl)-...)Copy SMILESCopy InChI

Affinity DataIC50: 170nMAssay Description:Antagonist activity against capsaicin-induced intracellular calcium ion increase in CHO cells expressing human TRPV1 in FLIPR assayMore data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In Depth
Date in BDB:
11/10/2009
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