BDBM50181460 1,3-bis(4-bromophenyl)-5-phenylimidazolidine-2,4-dione::CHEMBL383287

SMILES Oc1c(-c2ccccc2)n(-c2ccc(Br)cc2)c(=O)n1-c1ccc(Br)cc1

InChI Key InChIKey=KXPIARSCPWQBDY-UHFFFAOYSA-N

Data  2 KI  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 50181460   

TargetCannabinoid receptor 1(Human)
University of Louvain

Curated by ChEMBL
LigandPNGBDBM50181460(1,3-bis(4-bromophenyl)-5-phenylimidazolidine-2,4-d...)
Affinity DataEC50:  195nMAssay Description:Potency at human CB1 receptor in a [35S]GTP-gamma-S functional assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
University of Louvain

Curated by ChEMBL
LigandPNGBDBM50181460(1,3-bis(4-bromophenyl)-5-phenylimidazolidine-2,4-d...)
Affinity DataKi:  243nMAssay Description:Displacement of [3H]SR141716A from human CB1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2012
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Rat)
University of Louvain

Curated by ChEMBL
LigandPNGBDBM50181460(1,3-bis(4-bromophenyl)-5-phenylimidazolidine-2,4-d...)
Affinity DataKi:  311nMAssay Description:Displacement of [3H]SR141716A from CB1 receptor in rat cerebellumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2012
Entry Details Article
PubMed