BDBM50173303 CHEMBL3809560

SMILES Cn1cnc(Cn2nc3ccc(cn3c2=O)-c2ccc(OC(F)(F)F)cc2)n1

InChI Key InChIKey=PKMGMZYOIJAWBK-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50173303   

TargetSodium channel protein type 5 subunit alpha(Human)
Gilead Sciences

Curated by ChEMBL
LigandPNGBDBM50173303(CHEMBL3809560)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of 0.1 Hz stimulated human Nav1.5alpha expressed in HEK293 cells assessed as inhibition of late sodium current with 3 compound additions f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/7/2017
Entry Details Article
PubMed