BDBM50171235 5-Chloro-2-methyl-3-(1,2,3,6-tetrahydro-pyridin-4-yl)-1H-indole::CHEMBL364005

SMILES Cc1[nH]c2ccc(Cl)cc2c1C1=CCNCC1

InChI Key InChIKey=BPPGPYJBCVXILI-UHFFFAOYSA-N

Data  10 IC50  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 11 hits for monomerid = 50171235   

Target5-hydroxytryptamine receptor 6(Human)
Carlsson Research

Curated by ChEMBL
LigandPNGBDBM50171235(5-Chloro-2-methyl-3-(1,2,3,6-tetrahydro-pyridin-4-...)
Affinity DataIC50: 7.40nMAssay Description:Displacement of [3H]LSD binding to cloned human 5-hydroxytryptamine 6 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Carlsson Research

Curated by ChEMBL
LigandPNGBDBM50171235(5-Chloro-2-methyl-3-(1,2,3,6-tetrahydro-pyridin-4-...)
Affinity DataIC50: 240nMAssay Description:Inhibitory activity against 5-hydroxytryptamine 2A receptor in humanMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A(Human)
Carlsson Research

Curated by ChEMBL
LigandPNGBDBM50171235(5-Chloro-2-methyl-3-(1,2,3,6-tetrahydro-pyridin-4-...)
Affinity DataIC50: 34nMAssay Description:Inhibitory activity against 5-hydroxytryptamine 3 receptor expressed in NG 108 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Guinea pig)
Carlsson Research

Curated by ChEMBL
LigandPNGBDBM50171235(5-Chloro-2-methyl-3-(1,2,3,6-tetrahydro-pyridin-4-...)
Affinity DataIC50: 620nMAssay Description:Inhibitory activity against 5-hydroxytryptamine 4 receptor in guinea pigMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Carlsson Research

Curated by ChEMBL
LigandPNGBDBM50171235(5-Chloro-2-methyl-3-(1,2,3,6-tetrahydro-pyridin-4-...)
Affinity DataIC50: 660nMAssay Description:Inhibitory activity against 5-hydroxytryptamine 1A receptor in ratMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 7(Human)
Carlsson Research

Curated by ChEMBL
LigandPNGBDBM50171235(5-Chloro-2-methyl-3-(1,2,3,6-tetrahydro-pyridin-4-...)
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibitory activity against 5-hydroxytryptamine 7 receptor in humanMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Carlsson Research

Curated by ChEMBL
LigandPNGBDBM50171235(5-Chloro-2-methyl-3-(1,2,3,6-tetrahydro-pyridin-4-...)
Affinity DataIC50: 7.40nMAssay Description:Inhibitory activity against 5-hydroxytryptamine 6 receptor in humanMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1B(Rat)
Carlsson Research

Curated by ChEMBL
LigandPNGBDBM50171235(5-Chloro-2-methyl-3-(1,2,3,6-tetrahydro-pyridin-4-...)
Affinity DataIC50: 180nMAssay Description:Inhibitory activity against 5-hydroxytryptamine 1B receptor in ratMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1B(Human)
Carlsson Research

Curated by ChEMBL
LigandPNGBDBM50171235(5-Chloro-2-methyl-3-(1,2,3,6-tetrahydro-pyridin-4-...)
Affinity DataIC50: 110nMAssay Description:Inhibitory activity against 5-hydroxytryptamine 1B receptor in calfMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Human)
Carlsson Research

Curated by ChEMBL
LigandPNGBDBM50171235(5-Chloro-2-methyl-3-(1,2,3,6-tetrahydro-pyridin-4-...)
Affinity DataIC50: 450nMAssay Description:Inhibitory activity against 5-hydroxytryptamine 2C receptor in humanMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Carlsson Research

Curated by ChEMBL
LigandPNGBDBM50171235(5-Chloro-2-methyl-3-(1,2,3,6-tetrahydro-pyridin-4-...)
Affinity DataEC50:  1nMAssay Description:Partial agonist activity at 5-HT6 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2024
Entry Details
PubMed