BDBM50165195 CHEMBL3799946

SMILES Cc1noc(C)c1-c1cccc(COc2ccc(CCC(O)=O)c(F)c2)c1

InChI Key InChIKey=YZMQISQFDHASPC-UHFFFAOYSA-N

Data  3 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Similarity at least:  must be >=0.5
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 50165195   

TargetFree fatty acid receptor 1(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50165195(CHEMBL3799946)
Affinity DataEC50:  25nMAssay Description:Agonist activity at human GPR40 expressed in CHO cells by FLIPR calcium flux assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2017
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50165195(CHEMBL3799946)
Affinity DataEC50:  46nMAssay Description:Agonist activity at human FFA1 expressed in CHO cells assessed as increase in intracellular Ca2+ flux by Fluo-4 dye based FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50165195(CHEMBL3799946)
Affinity DataEC50:  33nMAssay Description:Agonist activity at human FFA1 receptor expressed in CHO cells assessed as increase in intracellular calcium levels measured for 1 hr by Fluo 4-AM dy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed