BDBM50163231 4-Pyridin-3-yl-piperazine-1-carboxylic acid (4-trifluoromethyl-phenyl)-amide::CHEMBL177003

SMILES FC(F)(F)c1ccc(NC(=O)N2CCN(CC2)c2cccnc2)cc1

InChI Key InChIKey=NAUBDHSOTWCGCF-UHFFFAOYSA-N

Data  1 IC50  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50163231   

TargetTransient receptor potential cation channel subfamily V member 1(Human)
Johnson & Johnson Pharmaceutical Research and Development

Curated by ChEMBL
LigandPNGBDBM50163231(4-Pyridin-3-yl-piperazine-1-carboxylic acid (4-tri...)
Affinity DataIC50: 5.03E+3nMAssay Description:Inhibition of human transient receptor potential vanilloid 1 receptor (n=3)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rat)
Johnson & Johnson Pharmaceutical Research and Development

Curated by ChEMBL
LigandPNGBDBM50163231(4-Pyridin-3-yl-piperazine-1-carboxylic acid (4-tri...)
Affinity DataEC50:  2.67E+3nMAssay Description:Effective concentration against rat transient receptor potential vanilloid 1 receptor (n=3)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed