BDBM50158897 CHEMBL3786105

SMILES FC(F)(F)c1ccc(C2CCOc3cc(ccc23)S(=O)(=O)Nc2nccs2)c(c1)C1=CCNCC1

InChI Key InChIKey=GUGZIAOSXOELAU-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50158897   

TargetSodium channel protein type 9 subunit alpha(Human)
Temple University

Curated by ChEMBL
LigandPNGBDBM50158897(CHEMBL3786105)
Affinity DataIC50: 1nMAssay Description:Inhibition of Nav1.7 (unknown origin) overexpressed in HEK293 cells preincubated for 15 to 20 mins followed by depolarization with 10 to 30 uM veratr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2017
Entry Details Article
PubMed