BDBM50157487 4-(6-hydroxy-1-propyl-1H-indazol-3-yl)benzene-1,3-diol::CHEMBL225514

SMILES CCCn1nc(-c2ccc(O)cc2O)c2ccc(O)cc12

InChI Key InChIKey=RJVVTFTZYVECEF-UHFFFAOYSA-N

Data  1 IC50  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50157487   

TargetEstrogen receptor(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50157487(4-(6-hydroxy-1-propyl-1H-indazol-3-yl)benzene-1,3-...)
Affinity DataEC50:  1.22E+3nMAssay Description:Activity at human ERalpha expressed in HAECT1 cells assessed as stimulation of creatine kinase activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEstrogen receptor(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50157487(4-(6-hydroxy-1-propyl-1H-indazol-3-yl)benzene-1,3-...)
Affinity DataIC50: 62nMAssay Description:Activity at human ERalpha expressed in HAECT1 cells assessed as inhibition of NF-kappaB transcriptionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed