BDBM50155652 3-Diethylamino-N-[6-(3-diethylamino-propionylamino)-9-oxo-9,10-dihydro-acridin-3-yl]-propionamide::CHEMBL1080436::CHEMBL362887

SMILES CCN(CC)CCC(=O)Nc1ccc2c(O)c3ccc(NC(=O)CCN(CC)CC)cc3nc2c1

InChI Key InChIKey=OZPBMVWVOOUJFN-UHFFFAOYSA-N

Data  1 IC50  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50155652   

TargetTelomerase reverse transcriptase(Human)
University of London

Curated by ChEMBL
LigandPNGBDBM50155652(CHEMBL1080436 | CHEMBL362887 | 3-Diethylamino-N-[6...)
Affinity DataEC50:  5.70E+3nMAssay Description:Concentration required to inhibit 50% of telomerase activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTelomerase reverse transcriptase(Human)
University of London

Curated by ChEMBL
LigandPNGBDBM50155652(CHEMBL1080436 | CHEMBL362887 | 3-Diethylamino-N-[6...)
Affinity DataIC50: 2.70E+3nMAssay Description:Inhibition of telomerase in human A2780 cells by TRAP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed