BDBM50155651 CHEMBL1081520::CHEMBL187955::N-[9-Oxo-6-(3-piperidin-1-yl-propionylamino)-9,10-dihydro-acridin-3-yl]-3-piperidin-1-yl-propionamide

SMILES Oc1c2ccc(NC(=O)CCN3CCCCC3)cc2nc2cc(NC(=O)CCN3CCCCC3)ccc12

InChI Key InChIKey=SIFRIGLNJULFCF-UHFFFAOYSA-N

Data  1 IC50  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Similarity at least:  must be >=0.5
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50155651   

TargetTelomerase reverse transcriptase(Human)
University of London

Curated by ChEMBL
LigandPNGBDBM50155651(CHEMBL1081520 | CHEMBL187955 | N-[9-Oxo-6-(3-piper...)
Affinity DataEC50:  5.90E+3nMAssay Description:Concentration required to inhibit 50% of telomerase activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTelomerase reverse transcriptase(Human)
University of London

Curated by ChEMBL
LigandPNGBDBM50155651(CHEMBL1081520 | CHEMBL187955 | N-[9-Oxo-6-(3-piper...)
Affinity DataIC50: 5.90E+3nMAssay Description:Inhibition of telomerase in human A2780 cells by TRAP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed