BDBM50155649 CHEMBL1078516::CHEMBL187202::N-[9-Oxo-7-(3-pyrrolidin-1-yl-propionylamino)-9,10-dihydro-acridin-2-yl]-3-pyrrolidin-1-yl-propionamide

SMILES Oc1c2cc(NC(=O)CCN3CCCC3)ccc2nc2ccc(NC(=O)CCN3CCCC3)cc12

InChI Key InChIKey=ZHGPGIWKJBAJMP-UHFFFAOYSA-N

Data  1 IC50  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50155649   

TargetTelomerase reverse transcriptase(Human)
University of London

Curated by ChEMBL
LigandPNGBDBM50155649(CHEMBL187202 | CHEMBL1078516 | N-[9-Oxo-7-(3-pyrro...)
Affinity DataEC50:  5.80E+3nMAssay Description:Concentration required to inhibit 50% of telomerase activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTelomerase reverse transcriptase(Human)
University of London

Curated by ChEMBL
LigandPNGBDBM50155649(CHEMBL187202 | CHEMBL1078516 | N-[9-Oxo-7-(3-pyrro...)
Affinity DataIC50: 5.80E+3nMAssay Description:Inhibition of telomerase in human A2780 cells by TRAP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed