BDBM50154237 CHEMBL187429::N-[4-(8-Benzhydryl-1,4-diaza-bicyclo[3.3.1]non-4-ylmethyl)-phenyl]-4-chloro-benzenesulfonamide

SMILES Clc1ccc(cc1)S(=O)(=O)Nc1ccc(CN2CCN3CC2CCC3C(c2ccccc2)c2ccccc2)cc1

InChI Key

Data  3 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 50154237   

TargetTransporter(Rat)
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50154237(N-[4-(8-Benzhydryl-1,4-diaza-bicyclo[3.3.1]non-4-y...)
Affinity DataIC50: 3.48E+3nMAssay Description:Inhibition of [3H]nisoxetine binding to norepinephrine transporter of rat cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50154237(N-[4-(8-Benzhydryl-1,4-diaza-bicyclo[3.3.1]non-4-y...)
Affinity DataIC50: 371nMAssay Description:Inhibition of [3H]WIN-35428 binding to dopamine transporter of rat striatumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Wayne State University

Curated by ChEMBL
LigandPNGBDBM50154237(N-[4-(8-Benzhydryl-1,4-diaza-bicyclo[3.3.1]non-4-y...)
Affinity DataIC50: 4.13E+3nMAssay Description:Inhibition of [3H]citalopram binding to serotonin transporter of rat cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2012
Entry Details Article
PubMed