BDBM50152031 7-(1-Cyclobutyl-ethyl)-3-(2,4-dichloro-phenyl)-8-ethyl-1-methyl-1,2,3,7-tetrahydro-purin-6-one::CHEMBL182068

SMILES CCc1nc2N(CN(C)C(=O)c2n1C(C)C1CCC1)c1ccc(Cl)cc1Cl

InChI Key InChIKey=VLFFGRQPWHSKJV-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50152031   

TargetCorticotropin-releasing factor receptor 1(Rat)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50152031(7-(1-Cyclobutyl-ethyl)-3-(2,4-dichloro-phenyl)-8-e...)
Affinity DataIC50: 26nMAssay Description:Inhibition of [125I]- Ovine CRF binding to rat frontal cortex corticotropin releasing factor 1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed