BDBM50143043 CHEMBL3758919

SMILES O=C1NC(=O)C(Cc2ccc(OCc3nc4ccccc4n3Cc3ccccc3)cc2)S1

InChI Key InChIKey=OGJMMQPQOZOCQR-UHFFFAOYSA-N

Data  2 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50143043   

TargetFree fatty acid receptor 1(Human)
Suez Canal University

Curated by ChEMBL
LigandPNGBDBM50143043(CHEMBL3758919)
Affinity DataEC50:  4.11E+3nMAssay Description:Agonist activity at human FFAR1 expressed in CHO-K1 cells assessed as calcium flux measured for 100 secs by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2017
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Suez Canal University

Curated by ChEMBL
LigandPNGBDBM50143043(CHEMBL3758919)
Affinity DataEC50:  3.02E+4nMAssay Description:Transactivation of N-terminal Gal4 DNA binding domain-linked human PPARalpha ligand binding domain after 24 hrs by luciferase reporter gene assay rel...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/8/2017
Entry Details Article
PubMed