BDBM50135587 CHEMBL335994::{(S)-5-Benzo[1,3]dioxol-5-yl-3-[(S)-3-(3,4-difluoro-phenyl)-2-methyl-propionylamino]-2-oxo-2,3-dihydro-benzo[e][1,4]diazepin-1-yl}-acetic acid methyl ester
SMILES COC(=O)CN1c2ccccc2C(=N[C@H](NC(=O)[C@@H](C)Cc2ccc(F)c(F)c2)C1=O)c1ccc2OCOc2c1
InChI Key InChIKey=DJNHHASAPQZIRO-UHFFFAOYSA-N
Data 1 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 50135587
TargetGamma-secretase subunit APH-1A/Gamma-secretase subunit APH-1B/Gamma-secretase subunit PEN-2/Nicastrin/Presenilin-1/Presenilin-2(Human)
Merck Sharp & Dohme Research Laboratories
Curated by ChEMBL
Merck Sharp & Dohme Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 13nMAssay Description:In vitro inhibition of gamma secretase.More data for this Ligand-Target Pair