BDBM50135576 (S)-N-[(S)-5-(2,2-Difluoro-benzo[1,3]dioxol-5-yl)-1-methyl-2-oxo-2,3-dihydro-1H-benzo[e][1,4]diazepin-3-yl]-3-(3,4-difluoro-phenyl)-2-methyl-propionamide::CHEMBL133235
SMILES C[C@@H](Cc1ccc(F)c(F)c1)C(=O)N[C@H]1N=C(c2ccc3OC(F)(F)Oc3c2)c2ccccc2N(C)C1=O
InChI Key InChIKey=WADIXAKIDBSZAJ-UHFFFAOYSA-N
Data 1 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 50135576
TargetGamma-secretase subunit APH-1A/Gamma-secretase subunit APH-1B/Gamma-secretase subunit PEN-2/Nicastrin/Presenilin-1/Presenilin-2(Human)
Merck Sharp & Dohme Research Laboratories
Curated by ChEMBL
Merck Sharp & Dohme Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 28nMAssay Description:In vitro inhibition of gamma secretase.More data for this Ligand-Target Pair